The organic chemistry of drug design and drug action /
Richard B. Silverman and Mark W. Holladay.
- Third edition.
- xviii, 517 pages : illustrations (some color) ; 29 cm
Includes bibliographical references and index.
Lead discovery and lead modification -- Receptors -- Enzymes -- Enzyme inhibition and inactivation -- DNA-interactive agents -- Drug resistance and drug synergism -- Drug metabolism -- Prodrugs and drug delivery systems.